Zepbound (Tirzepatide Injection)

Name: Zepbound
Brand: Eli Lilly
SKU: 7821
Availability: InStock

Type

Product

Manufacturer

Country

Dosage

Qty-Price (USD)

Type:

Product: Zepbound 2.4ml kwikPen Pre-filled Pen (Local Pick-UP Only)

Manufacturer: Eli Lilly

Country: Canada

Dosage: 2.5 mg/0.6 ml

Qty-Price (USD):

Type:

Product: Zepbound 2.4ml kwikPen Pre-filled Pen (Local Pick-UP Only)

Manufacturer: Eli Lilly

Country: Canada

Dosage: 5 mg/0.6 ml

Qty-Price (USD):

Type:

Product: Zepbound 2.4ml kwikPen Pre-filled Pen (Local Pick-UP Only)

Manufacturer: Eli Lilly

Country: Canada

Dosage: 7.5 mg/0.6 ml

Qty-Price (USD):

Type:

Product: Zepbound 2.4ml kwikPen Pre-filled Pen (Local Pick-UP Only)

Manufacturer: Eli Lilly

Country: Canada

Dosage: 10 mg/0.6 ml

Qty-Price (USD):

Type:

Product: Zepbound 2.4ml kwikPen Pre-filled Pen (Local Pick-UP Only)

Manufacturer: Eli Lilly

Country: Canada

Dosage: 12.5 mg/0.6 ml

Qty-Price (USD):

Generic Equivalent of Zepbound

Type

Product

Manufacturer

Country

Dosage

Qty-Price (USD)

There is no generic product of Zepbound.

Zepbound Information

Tirzepatide injection at CanadaPharmacyOnline.com

The manufacturer of brand-name Zepbound (tirzepatide) is Eli Lilly and Company. Zepbound is a revolutionary, dual-action injectable medication approved for chronic weight management. It contains the same active ingredient as Mounjaro, which is used for type 2 diabetes, but Zepbound is specifically indicated for obesity and weight-related conditions.

The generic tirzepatide injection is currently unavailable at this pharmacy.

Dosage:

Zepbound is available in the following strengths, delivered via a single-dose pre-filled pen:
• Pre-filled Pen: 2.5 mg, 5 mg, 7.5mg, 10 mg, and 12.5 mg in 0.6 ml KwikPen

The dosage will be increased incrementally based on your weight-loss progress and tolerability.

Usage:

Zepbound is used for chronic weight management in adults with obesity (BMI of 30 kg/m3), overweight (BMI of 27 kg/m3 or greater) who also have at least one weight-related condition, such as high blood pressure, type 2 diabetes, or high cholesterol. Zepbound was recently approved for adults with moderate-to-severe OSA and obesity to improve sleep symptoms.

Mechanism of Action
Tirzepatide, the active ingredient in Zepbound, is a dual agonist that mimics two natural hormones. It is a GLP-1 (glucagon-like peptide-1) agonist that targets the brain to reduce hunger and slows stomach emptying, making you feel full longer. It also acts as a GIP (glucose-dependent insulinotropic polypeptide) agonist, further improving the body's breakdown of sugar and fat. By activating both pathways simultaneously, Zepbound provides a more powerful signal to the brain's reward and appetite centers than single-hormone drugs, often resulting in more significant weight loss.

Take Zepbound exactly as your doctor prescribes, according to the product monograph. Administer once weekly, at any time of day, with or without meals. Inject subcutaneously (under the skin) in the abdomen, thigh, or back of the upper arm. Rotate your injection site each week.

The information below summarizes some, but not all, potential side effects, risks, and interactions. Before starting Zepbound, it is essential to discuss all possible side effects, risks, and interactions with your doctor or pharmacist.

Side Effects:

The information below outlines potential side effects of Zepbound (tirzepatide injection). It is not an exhaustive list, and individual reactions can vary.

Common side effects: These are common side effects of Zepbound; other side effects are possible. Contact your doctor promptly if any side effects are persistent, worsening, or concerning, or if you experience any other concerning symptoms.
• Constipation
• Diarrhea
• Fatigue
• Heartburn
• Nausea
• Vomiting

Serious Side Effects: Seek immediate medical attention or call emergency services if you experience any of the following symptoms:
• Gallbladder Problems: Pain in the upper right stomach, fever, or yellowing of the skin/eyes.
• Kidney Issues: Severe dehydration from vomiting/diarrhea can lead to kidney failure.
• Severe Abdominal Pain: Could be a sign of pancreatitis (inflammation of the pancreas).
• Suicidal Thoughts: Pay attention to any sudden changes in mood or behavior.

Contraindications:

The following is not an exhaustive list of contraindications. Before starting Zepbound, it is crucial to discuss all your medical conditions, past and present, and all medications you are taking with your doctor or pharmacist.

Do not take Zepbound/tirzepatide injection if:
• Allergies: You have a known hypersensitivity to tirzepatide or any of its ingredients.
• Thyroid Cancer Risk: Do not use if you or your family have a history of Medullary Thyroid Carcinoma (MTC) or Multiple Endocrine Neoplasia syndrome type 2 (MEN 2).

Tell your doctor about all of your medical conditions, past and present, before starting Zepbound. This is crucial as certain conditions affect the drug's safety.
• Pregnancy: Zepbound is not recommended during pregnancy and should be stopped at least 2 months before a planned pregnancy.
• Severe Stomach Issues: Use with caution if you have severe gastroparesis (slowed stomach emptying).

Drug Interactions:

Before taking Zepbound, discuss all potential risks and interactions with your doctor or pharmacist. For complete and up-to-date information, please visit the prescribing information at https://pi.lilly.com/us/zepbound-uspi.pdf.

Provide your doctor with a complete list of all your medications, including prescriptions, over-the-counter (OTC) drugs, vitamins, herbal supplements, recreational drugs, and any significant dietary changes, as these may interact with Zepbound. Zepbound may interact with other medicines, including but not limited to:
• Oral Contraceptives: Zepbound slows stomach emptying, which may affect how birth control pills are absorbed. Your doctor may recommend a non-oral or backup method for 4 weeks after starting and after each dose increase.
• Insulin and Sulfonylureas: Taking Zepbound with these can increase the risk of dangerously low blood sugar (hypoglycemia).

Pregnancy and Breastfeeding:

Zepbound is not recommended during pregnancy. Weight loss is generally not advised for pregnant individuals, as it can harm fetal development. If you are planning to become pregnant, experts recommend stopping Zepbound at least 2 months before trying to conceive to ensure the medication has fully cleared your system. It is currently not known if tirzepatide passes into human breast milk or how it might affect a nursing infant. Because the risks are unclear, you should discuss the benefits and potential risks with your doctor before using Zepbound while nursing.

Use in Children:

The safety and effectiveness of Zepbound in children and adolescents under 18 years of age have not yet been established.

Frequently Asked Questions about Zepbound at Canada Pharmacy Online

Why is Zepbound more affordable in Canada than in the United States?

Prescription drug prices, including Zepbound, are generally lower in Canada than in the U.S. due to a combination of factors, primarily government price regulations, differing market dynamics, and other economic considerations. In Canada, provincial and federal governments negotiate drug prices with pharmaceutical companies, which often results in lower prices than in the U.S., where market forces play a more significant role. For more information, see the FAQs on Prescription Drug Importation from the Kaiser Family Foundation (KFF): https://www.kff.org/health-costs/issue-brief/faqs-on-prescription-drug-importation/

How much is the shipping?

Our shipping fee is a flat rate of $10.00 per order. Our pharmacy is dedicated to offering you the lowest prices on high-quality products.

How do I place an order with your pharmacy?

Ordering from us is very simple. You can purchase online or call Customer Service at 1866.920.3784; for more information or to learn about the ordering process, visit our How to Order page.

Is there a limit on how many Zepbound Injection I can order at once?

CanadaPharmacyOnline.com can dispense up to a three-month supply of Zepbound per prescription from your doctor.

Can I buy Zepbound from you over the counter?

No, Zepbound requires a valid prescription from your doctor. We do not sell this product without a valid prescription.

Do you ship to the United States?

Yes, we do. It usually takes between 7 and 18 business days to receive your order from our pharmacy.

Is there a generic for Zepbound?

No, the generic tirzepatide injection is currently unavailable (at this pharmacy).

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The information on this page is sourced from independent third parties contracted by CanadaPharmacyOnline. While we cannot guarantee its medical accuracy, we strongly recommend consulting a healthcare professional for personalized advice regarding medications or medical conditions.

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