Isentress (Raltegravir)

Name: Isentress
Brand: Merck
SKU: 6558
Availability: InStock

Type

Product

Manufacturer

Country

Dosage

Qty-Price (USD)

Type:

Product: Isentress Chew Tablet

Manufacturer: Merck

Country: Canada

Dosage: 25 mg

Qty-Price (USD):

Type:

Product: Isentress Chew Tablet

Manufacturer: Merck

Country: Canada

Dosage: 100 mg

Qty-Price (USD):

Type:

Product: Isentress

Manufacturer: Merck

Country: Canada

Dosage: 400 mg

Qty-Price (USD):

Type:

Product: Isentress

Manufacturer: Merck

Country: India

Dosage: 400 mg

Qty-Price (USD):

Type:

Product: Isentress HD Tablet

Manufacturer: Merck

Country: Canada

Dosage: 600 mg

Qty-Price (USD):

Generic Equivalent of Isentress

Type

Product

Manufacturer

Country

Dosage

Qty-Price (USD)

Type:

Product: Raltegravir (Cipla-Zepdon)

Manufacturer: Generic

Country: India

Dosage: 400 mg

Qty-Price (USD):

Isentress Information

Isentress and Raltegravir at CanadaPharmacyOnline.com

Brand Isentress (raltegravir) is manufactured by Merck in many countries worldwide, including Canada and India.

Generic raltegravir is sourced from manufacturers that meet applicable regulatory standards. The specific manufacturer of your dispensed medication may vary.

Important Information about Generic Raltegravir:

Generic raltegravir contains the same active ingredient as the brand-name Isentress. It must meet the same safety, effectiveness, and quality standards as the brand-name product. This means it is designed to work in the same way as Isentress. Studies have demonstrated bioequivalence between generic and brand-name raltegravir, indicating comparable absorption rates and overall effects. However, individual responses to any medication can vary. If you have any questions about using generic raltegravir, talk to your doctor or pharmacist.

For more information about generic drug approval and bioequivalence, you can visit the FDA website: https://www.fda.gov/drugs/buying-using-medicine-safely/generic-drugs

Dosage:

Isentress is commonly available in different forms and dosages, including:
• 25 mg and 100 mg chewable tablets
• 400 mg and 600 mg film-coated tablets

The generic raltegravir is also available as 400 mg oral tablets.

Your doctor will determine the appropriate dose based on your individual needs and medical conditions.

Usage:

Isentress (raltegravir) is a prescription medication primarily used to treat HIV-1 infection in adults and children. It is used as part of combination antiretroviral therapy and is not taken alone. HIV attacks the immune system, weakening the body's ability to fight infections. Isentress does not cure HIV, but when taken consistently with other HIV medicines, it lowers the amount of virus in the blood, helps protect the immune system, and reduces the risk of HIV-related illness and transmission.

Mechanism of Action:
Isentress (raltegravir) is an integrase strand transfer inhibitor (INSTI). It works by blocking the HIV integrase enzyme, which the virus needs to insert its genetic material into human immune cells. Without this step, HIV cannot successfully reproduce. By stopping viral replication early in its life cycle, Isentress helps control HIV infection when used with other antiretroviral drugs.

Take Isentress exactly as your doctor prescribes, following the instructions in the product monograph in Canada that accompanies the medication. Consult your doctor for personalized guidance and safe use.

The information below summarizes some, but not all, potential side effects, risks, and interactions. Before taking Isentress, it is essential to discuss all possible side effects, risks, and interactions with your doctor or pharmacist.

Side Effects:

The information below outlines potential side effects associated with Isentress (raltegravir). It is not an exhaustive list, and individual reactions can vary. This information is for educational purposes and should not replace professional medical advice. Before starting Isentress, it is crucial to discuss possible side effects and risks with your doctor or pharmacist.

Common side effects - These are common side effects of Isentress; others are possible. Contact your doctor promptly if any side effects persist, worsen, or concern you, or if you experience any other concerning symptoms.
• Diarrhea
• Headache
• Nausea
• Sleeping difficulties
• Stomach pain
• Tiredness

Serious or rare side effects- Seek immediate medical attention or call emergency services if you experience any of the following:
• Severe skin reactions with peeling or blistering;
• Signs of an allergic reaction, such as swelling, breathing difficulties, swelling of the face, lips, or throat;
• Signs of liver problems, including yellowing of the skin or eyes, dark urine;
• Signs of possible muscle injury, including muscle pain, weakness, or dark urine

Contraindications:

The following is not an exhaustive list of contraindications. Before starting Isentress, it is essential to discuss all your medical conditions, past and present, as well as all medications you are currently taking, with your doctor or pharmacist.

Isentress should not be used if:
• You have a known allergy to raltegravir or any of the ingredients in the medication

Tell your doctor about all of your medical conditions, past and present, before starting Isentress. This is crucial because certain conditions can affect whether Isentress is right for you. These conditions may include, but are not limited to:
• Kidney disease
• Liver disease, including hepatitis B or C
• Muscle disorders

Drug Interactions:

Before taking Isentress, it is essential to discuss all potential risks and interactions with your doctor or pharmacist. For complete and up-to-date information, please visit the patient medication information from Merck Canada at https://www.merck.ca/en/wp-content/uploads/sites/20/2021/04/ISENTRESS-CI_E.pdf.

Provide your doctor with a complete list of all your medications, including prescriptions, over-the-counter (OTC) drugs, vitamins, and herbal supplements. It is also essential to inform your doctor about any herbal teas, recreational drugs, or significant dietary changes you are making, as these could potentially interact with Isentress. Isentress may interact with other medicines, but is not limited to:
• Aluminum and magnesium-based antacids – should not be taken with Isentress because they significantly reduce the medication's absorption. While not listed as an official contraindication, co-administration is not recommended by the manufacturer.
• Other HIV medications – Some combinations require dose adjustments when used with Isentress. Your doctor will review your HIV regimen as a whole.
• Other strong enzyme inducers, such as certain seizure medications, may reduce raltegravir's effectiveness.
• Rifampin – Can lower raltegravir levels, potentially reducing HIV control.

Pregnancy and Breastfeeding:

Isentress may be used during pregnancy. Your doctor will prescribe the medicine if the benefits outweigh the risks. Breastfeeding is now supported by the WHO and many national health agencies for mothers living with HIV, provided they maintain a sustained undetectable viral load on antiretroviral therapy (ART). The risk of HIV transmission through breastfeeding is negligible—effectively zero—provided the mother maintains a sustained undetectable viral load on antiretroviral therapy (ART). Consult your doctor for the most current clinical management guidelines.

Frequently Asked Questions about Isentress at Canada Pharmacy Online:

Why is Isentress more affordable in Canada than in the United States?

Prescription drug prices, including Isentress, are generally lower in Canada than in the U.S. due to a combination of factors, primarily government price regulations, differing market dynamics, and other economic considerations. In Canada, provincial and federal governments negotiate drug prices with pharmaceutical companies, which often results in lower prices than in the U.S., where market forces play a more significant role. For more information, see the FAQs on Prescription Drug Importation from the Kaiser Family Foundation (KFF): https://www.kff.org/health-costs/issue-brief/faqs-on-prescription-drug-importation/

How much is the shipping?

Our shipping fee is a flat rate of $10.00 per order. Our pharmacy is dedicated to providing you with the lowest prices on high-quality products.

How do I place an order with your pharmacy?

Ordering from us is very simple. You can purchase online or call Customer Service at 1866.920.3784; for more information or to learn about the ordering process, visit our How to Order page.

Is there a limit on the number of tablets I can order at one time?

CanadaPharmacyOnline.com can only dispense a maximum of a three-month supply of Isentress at a time, as per your doctor's prescription.

Can I buy over the counter from you?

No, Isentress requires a valid prescription from your doctor. We do not sell this product without a valid prescription.

Do you ship to the United States?

Yes, we do. It typically takes 7-18 business days for your order to be delivered from our pharmacy.

Is Isentress a cure for HIV?

No. Isentress controls HIV but does not cure it. Daily adherence is essential.

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The information on this page is sourced from independent third parties contracted by CanadaPharmacyOnline. While we cannot guarantee its medical accuracy, we strongly recommend consulting a healthcare professional for personalized advice regarding medications or medical conditions.

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